Obviously, the structure and function of receptors is a complex science and is, understandably, a casual interest for most of us. Certain principles have significant clinical value, however. If the general effects of specific receptors are understood, one can predict the indications and effects of many drugs used in clinical practice. For example, beta receptors in the heart mediate excitatory events. Drugs acting as agonists at beta receptors increase heart rate and are used to manage bradycardia. Conversely, beta-receptor antagonists decrease heart rate and can be used